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Bantag-1 trifluoroacetate
CAS No. ——
Bantag-1 trifluoroacetate( —— )
Catalog No. M17037 CAS No. ——
A potent, highly selective, peptide bombesin receptor subtype-3 (BRS-3) antagonist with IC50 of 2-8 nM for human and rodent BRS-3.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
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Biological Information
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Product NameBantag-1 trifluoroacetate
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NoteResearch use only, not for human use.
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Brief DescriptionA potent, highly selective, peptide bombesin receptor subtype-3 (BRS-3) antagonist with IC50 of 2-8 nM for human and rodent BRS-3.
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DescriptionA potent, highly selective, peptide bombesin receptor subtype-3 (BRS-3) antagonist with IC50 of 2-8 nM for human and rodent BRS-3, displays 1000-fold selectivity over hNMBR and hGRPR, increases food intake and produces an obesity phenotype in mice.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayGPCR/G Protein
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TargetBombesin Receptor
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RecptorBombesin Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number——
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Formula Weight——
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Molecular FormulaC48H73N8O7 · xC2HF3O2
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Purity>98% (HPLC)
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Solubility——
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SMILES——
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Chemical NameBoc-Phe-His-4-amino-5-cyclohexyl-2,4,5-trideoxypentonyl-Leu-(3-dimethylamino) benzylamide N-methylammonium trifluoroacetate salt
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Moreno P, et al. J Pharmacol Exp Ther. 2013 Oct;347(1):100-16.
2. Guan XM, et al. Cell Metab. 2010 Feb 3;11(2):101-12.
3. Feng Y, et al. Endocrinology. 2011 Nov;152(11):4106-15.
4. Nakamura T, et al. Biochem Pharmacol. 2016 Sep 1;115:64-76.
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